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PNASM- Production scientifique 2014-15


18 - Small molecules inhibitors of plasminogen activator inhibitor-1 – An overview. A. Rouch, C. Vanucci-Bacqué, F. Bedos-Belval, M. Baltas. Eur. J. Med. Chem., 2015, 92, 619-636.

17 - Crystal structure of the enoyl-ACP reductase of Mycobacterium tuberculosis (InhA) in the apo-form and in complex with the active metabolite of isoniazid pre-formed by a biomimetic approach. A. Chollet, L. Mourey, C. Lherbet, A. Delbot, S. Julien, M. Baltas, J. Bernadou, G. Pratviel, L. Maveyraud, V. Bernardes-Génisson. J. Struct. Biol. 2015, 190, 328-337.

16 - Synthesis and evaluation of a-hydroxytriazoles and related compounds as antitubercular agents. C. Menendez, G. Mori, M. Maillot, I. Fabing, C. Carayon, B.S. Orena, M.R. Pasca, Z. Voitenko, C. Lherbet, M. Baltas. French-Ukrain. J. Chem. 2015, 3, 82-96.

15 - Design, synthesis and evaluation of new GEQ derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis. A. Chollet, G. Mori, C. Menendez, F. Rodriguez, I. Fabing, M.R. Pasca J. Madacki, J. Kordulakova, P. Constant, A. Quémard, V. Bernardes-Génisson, M. Baltas.  Eur. J. Med. Chem. 2015, 101, 218-235

14 - Two new metal-organic framework structures derived from terephthalate and linear trimetallic zinc building units N. Saffon-Merceron, M.C. Barthelemy, C. Laurent, I. Fabing, P. Hoffmann, A. Vigroux. Inorganica Chimica Acta, 2015, 426, 15-19.


13 - The first example of an unusual rearrangement in the van Leusen imidazole synthesis. M. Fodili, B. Nadjar-Kolli, M. Vedrenne, N. Saffon-Merceron, C. Lherbet, P. Hoffmann. Chem. Heterocycl. Compd. 2015, 51, 940-943.


12 - Synthesis and in vitro antiproliferative activities of amido- and amino-analogues of the marine alkaloid isogranulatimide. B. Salvetti, H. Lavrard, V. Mathieu, F. Rodriguez, R. Kiss, E. Delfourne. Chem. Med. Chem. 2015, 10, 607-609.


11 - Unexpected copper mediated benzyl O->O migration during an Ulmann ether coupling. C. Vanucci-Bacqué, S. Chaabouni, I. Fabing, F. Bedos-Belval, M. Baltas. Tetrahedron Lett., 2014, 55, 528-530.


10 - Synthesis, antioxidant and cytoprotective evaluation of potential antiatherogenic phenolic hydrazones. A structure-activity relationship insight. C. Vanucci-Bacqué,Ch. Carayon, C. Bernis, C. Camare, A. Nègre-Salvayre, F.Bedos-Belval, M. Baltas. Bioorg. Med. Chem. 2014, 22, 4269-4276.


9 - Reductive dimerization mechanisms of some streptocyanine dyes. C. André-Barrès, F. Najjar, M.-P. Maether, C. Payrastre, T. Tzedakis, P. Winterton. Electrochimica Acta 2014, 132, 423-433.

8 - Antimalarial bicyclic peroxides belonging to the G-factor family: mechanistic aspects of their formation and iron (II) induced reduction. J. Ruiz, J. Azéma, C. Payrastre, M. Baltas, B. Tuccio, H. Vial, C. André-Barrès. Current Topics in Medicinal Chemistry, 2014, 14,1668-1683.

7 - Design, synthesis and evaluation of new tricyclic endoperoxides as potential antiplsamodial agents. J. Ruiz, S. Ladeira, H. Vial, C. André-Barrès. Org. Biomol. Chem., 2014, 28, 5212-5221.

6- Design of granulatimide and isogranulatimide analogues as potential Chk1 inhibitors: study of amino-platforms for their synthesis. H. Lavrard, F. Rodriguez, E. Delfourne. Bioorg. Med. Chem. 2014, 22, 4961-4967.

5 - Synthesis of substituted amido-isogranulatimide analogues as potent checkpoint kinase inhibitors. B. Salvetti, H. Lavrard, E. Delfourne. Tetrahedron Lett. 2014, 55, 6463-6464.

4 - Synthesis of 3-heteryl substituted pyrrolidine-2,5-diones via catalytic Michael reaction and evaluation of their inhibitory activity against InhA and Mycobacterium tuberculosis. T. Matviiuk, G. Mori, C. Lherbet, F. Rodriguez, M.R. Pasca, M. Gorichko, B. Guidetti, Z. Voitenko, M. Baltas. Eur. J. Med. Chem. 2014, 71, 46-52.

3 - Solvent-free mechanochemical route for green synthesis of pharmaceutically attractive phenol-hydrazones. F. Oliveira, M. Baron, A. Chamayou, C. Andre-Barres, B. Guidetti, M. Baltas. RSC Advances, 2014, 4, 56736-56742.


2 - Synthesis of alpha-Keto-1,2,3-triazoles through copper iodide catalyzed oxygenation. S. Nawratil, M. Grypioti, C. Menendez, S. Mallet-Ladeira, C. Lherbet, M. Baltas. Eur. J. Org. Chem, 2014, 3, 654-659.

1 - LiAlH4 promoted tandem reduction/oxidation of fluorenyl derivatives under air. T. Matviiuk, C. Menendez, C. Carayon, N. Saffon,  Z. Voitenko, C. Lherbet, M. Baltas.  Eur. J. Org. Chem, 2014, 29, 6538-6546.


Date de mise à jour 29 novembre 2017


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