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26 sept.

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PNASM- Production scientifique 2016-17

25- Synthesis, biological evaluation and in silico molecular modeling of pyrrolyl benzohydrazide derivatives as enoyl ACP reductase inhibitors.
S.D. Joshi, S.R. Dixit, V.H. Kulkarni, C. Lherbet, M.N. Nadagouda, T.M. Aminabhavi
Eur. J. Med. Chem., 2017, 126, 286-297.

24 – Comprehensive experimental investigation of mechanically induced 1,4-diazines synthesis in solid state
P.F.M. Oliveira, N. Haruta, A. Chamayou, B. Guidetti, M. Baltas , K. Tanaka, T. Sato, M. Baron
Tetrahedron, 2017, 73, 2305–2310.

23- New reaction of formation of the fused tricyclic bispyrroloquinone ring system
A. Vanicat,  C. André-Barrès, E. Delfourne
Tetrahedron Lett., 2017, 58,  342–345.

22 – Total Synthesis of Tedarene A
K. Maurent, C. Vanucci-Bacque, N. Saffon-Merceron, M. Baltas, F. Bedos-Belval
J.  Nat. Prod., 2017, 80, 1623-1630.

21 – Insights into Substrate Modification by Dehydratases from Type I Polyketide Synthases
A. Faille, S. Gavalda, N. Slama, C. Lherbet, L. Maveyraud, V. Guillet, F. Laval, A. Quemard,  L. Mourey, J.D Pedelacq
J. Mol. Biol., 2017, 429, 1554-1569. 

20 – A revisited structure for nitrosoprodenafil from NMR, mass spectrometry, X-ray and hydrolysis data
R. Martino, C. Menendez, S. Balayssac, N. Martins-Froment, C. Lherbet, F. Couderc, V. Gilard, M. Malet-Martino
J.  Pharm. Biomed. Anal., 2017, 135, 31-49.

19- 4-Hydroxynonenal contributes to angiogenesis through a redox-dependent sphingolipid pathway. Prevention by hydralazine derivatives. Camaré C., Auge N., Vanucci-Bacqué C., Pucelle M., Bernis C., Swiader A., Baltas M., Bedos-Belval F., Salvayre R. S., Negre-Salvayre A.
Oxid. Med. Cell Longev, 2017, 9, 1-11.

18-Mechanochemical Synthesis and Biological Evaluation of Novel Isoniazid Derivatives with Potent Antitubercular Activity
Oliveira P. F. M., Guidetti B., Chamayou A. et al.
Molecules, 2017, 22, 1457-1484.

17 - Hemisynthesis, Antitumoral Effect, and Molecular Docking Studies of Ferutinin and Its Analogues.
R. Safi, F. Rodriguez, G. Hilal, M. Diab-Assaf, Y. Diab, M. El-Sabban, F. Najjar, E. Delfourne
Chem. Biol. Drug Des., 2016, 87, 382-397. 

16 - Antioxidant activity of a series of amides
F. Malki, A. Touati, K. Hamza, S. Moulay, M. Baltas
J. Mater. Environ. Sci., 2016, 7, 936-941.

15 - Antioxydant and antimicrobial activities of two amidine derivatives
F. Malki, A. Touati, S. Moulay, M. Baltas
Mediterr. J. Bio., 2016, 1, 62-68.

14 – Structure-Based Virtual Ligand Screening on the XRCC4/DNA Ligase IV Interface
G. Menchon, O. Bombarde, M. Trivedi, A. Négrel, C. Inard, B. Guidetti, M. Baltas, A. Milon, M. Modesti, G. Czaplicki, P. Calsou
Nature, Scientific Reports, 2016, 6, 22878.

13 – Design, synthesis and biological evaluation of novel hydroxamic acids  bearing artemisinin skeleton
V. T. Ha, V. T.Kien, L. H. Binh, V. D. Tien, Nguyen T. T. My, Nguyen Hai Nam, M. Baltas, H. Hahn, B. Woo Han, D. Thi Thao, T. Khac Vu
BioOrg. Chem
., 2016, 66, 63–71.

12 - Triazolophthalazines - Easily Accessible Compounds with Potent Antitubercular Activity
D Veau,  S. Krykun, G. Mori, B. S. Orena, M. R. Pasca, C. Frongia, V. Lobjois, S. Chassaing, C. Lherbet and M. Baltas
Chem. Med. Chem, 2016, 11, 1078-1089

11 – Identification and optimization of hydrazine-gallate derivatives as specific inhibitors of DNA methyltransferase 3A
A. Erdmann, Y. Menon, C. Gros, V. Masson, Y.Aussagues, F. Ausseil, N. Novosad, P. Schambel, M. Baltas, & P.B. Arimondo
Future Med. Chem., 2016, 8, 373-380.

10 - Lowering the Activation Energy under Mechanochemical Conditions: The Case of 2,3-diphenylquinoxaline
P. F. M. Oliveira, M. Baron, A. Chamayou, M. Baltas, B. Guidetti, N. Haruta, K. Tanaka, T. Sato
ChemistrySelect, 2016, 5, 984-988.

9 - Peptide Synthesis in Ionic Liquids (PEPSIL): All You Need is in the Toolbox!
K. Jebri, N. Galy, V. Zgonnik, M.R. Mazières, Y. Génisson, F. Guillen, T.B. Ayed, M. Baltas, J.C. Plaquevent
French-Ukrain. J.  Chem., 2016, 4, 3-13.

8 – Synthesis and evaluation of antioxidant phenolic diaryl hydrazones as potent antiangiogenic agents in atherosclerosis
C. Vanucci-Bacqué, C. Camare, C. Carayon, C. Bernis, M. Baltas, A. Nègre-Salvayre, F. Bedos-Belval
Biorg. Med.Chem., 2016, 24, 3571-3578

7 -Synthesis, characterization and antitubercular activities of novel pyrrolyl hydrazones and their Cu-complexes
D. Kumar, S.R. Dixit, N. Tigadi, U.A. More, C. Lherbet, T.M. Aminabhavi, K.S Yang
Eur. J. Med. Chem. 2016, 121, 21-39.

6 - Synthesis, antimycobacterial screening and ligand-based molecular docking studies on novel pyrrole derivatives bearing pyrazoline, isoxazole and phenyl thiourea moieties
S.R Dixit, Kirankumar M N, T.M Aminabhavi, K. V. S. N. Raju, R. Narayan, C. Lherbet, K.S. Yang, S. Joshi
Eur. J. Med. Chem. 2016, 107, 133-152

5 - Pyrrolidinone and pyrrolidine derivatives: Evaluation as inhibitors of InhA and Mycobacterium tuberculosis
T. Matviiuk,  J. Madacki,  G. Mori, B. Silvia Orena, C. Menendez,  A. Kysil, C. André-Barrès, F. Rodriguez, J. Korduláková, S. Mallet-Ladeira,  Z. Voitenko, M.R. Pasca,  C. Lherbet, M. Baltas
Eur. J. Med. Chem. 2016, 123, 462-475

4 –An Unusual 3D Zinc Organic Framework Constructed from Paddle Wheel Based Carboxylate Sheets Pillared by Nitrate Ions.
N. Saffon-Merceron, C. Laurent, I. Fabing, P. Hoffmann, A. Vigroux
 Z. Anorg. Allg. Chem. 2016, 642, 709-713.

3 - An Unexpected Reaction of 3-Ethoxycyclohex-2-enone with 3-Oxo-1,2-pyrazolidinium ylides: Preparation of 9-aryl-xanthenediones
O. Amiri, N. Belkhouya, M. Alaoui, S. Mojahidi, L. Bouissane, M. Baltas, R. Brousse, and E.M. Rakib
Der Pharm. Chem., 2016, 8, 1-5.

2 - Evaluation of the inhibitory activity of (aza)isoindolinone-type compounds: toward in vitro InhA action, Mycobacterium tuberculosis growth and mycolic acid biosynthesis.
A. Chollet, J.L. Stigliani, M.R. Pasca, G. Mori, C. Lherbet, P. Constant, A. Quemard, J. Bernadou, G. Pratviel,V. Bernardes-Genisson
Chem. Biol. & Drug Des., 2016, 88, 740-755.

1 – Novel artemisinin-derived dimers: synthesis and evalution of anticancer activities.
Vu Tuan Kien, Le Huy Binh, Phan hai Phong, Doan Thi Hien, Nguyen Thi Thuy My, Nguyen Hai Nam, Do Thi Thao, Michel Baltas, Tran Khac Vu
Lett. Drug Des. Discov., 2016, 13, 1-10





Date de mise à jour 30 novembre 2017


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